Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM270279((2S,3R)-3-(3-(((S)-1-(2,5-bis(trifluoromethyl)benz...)
BDBM270279((2S,3R)-3-(3-(((S)-1-(2,5-bis(trifluoromethyl)benz...)
BDBM270279((2S,3R)-3-(3-(((S)-1-(2,5-bis(trifluoromethyl)benz...)
EC50: 51nMpH: 7.4 T: 2°CAssay Description:FLIPR (Fluorimetric Imaging Plate Reader, Molecular Devices) assays were performed to measure agonist-induced calcium mobilization of the stable clon...More data for this Ligand-Target Pair
BDBM270279((2S,3R)-3-(3-(((S)-1-(2,5-bis(trifluoromethyl)benz...)
EC50: 89nMT: 2°CAssay Description:The assay was performed in 96-well format. HEK cells stably expressing human GPR40 were plated to be 60-80% confluent within 72 h. After 72 h, the pl...More data for this Ligand-Target Pair