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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at Gal4-fused human PPAR-alpha ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-gamma ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  24nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  3.70E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-alpha ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at Gal4-fused human PPAR-gamma ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed