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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Platelet glycoprotein 4
(Rattus norvegicus)
Valorisation-Recherche, Limited Partnership
US Patent
Ligand
BDBM263256
(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)
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Affinity Data
IC50: 2.95E+3nM
pH: 7.3
Assay Description:
Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
US Patent
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Target
Platelet glycoprotein 4
(Rattus norvegicus)
Valorisation-Recherche, Limited Partnership
US Patent
Ligand
BDBM263256
(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)
Copy SMILES
Affinity Data
IC50: 9.19E+3nM
Assay Description:
Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysis
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Estrogen receptor [D538G]
(Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership
US Patent
Ligand
BDBM263256
(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)
Copy SMILES
Affinity Data
IC50: 1.00E+4nM
Assay Description:
GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI