Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Cytosol aminopeptidase
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 290nM
Assay Description:
Inhibition against Leucyl aminopeptidase from pig kidney.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro aminopeptidase 2
(Rattus norvegicus)
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 660nM
Assay Description:
Activity against membrane bound rat aminopeptidase P
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro aminopeptidase 1
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.70E+3nM
Assay Description:
Inhibition against cytosolic Aminopeptidase P from human heart.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro aminopeptidase 2
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.80E+3nM
Assay Description:
Inhibition against membrane bound human aminopeptidase P
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro aminopeptidase 2
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.40E+3nM
Assay Description:
Inhibition against membrane bound monkey aminopeptidase P
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro aminopeptidase 1
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.80E+3nM
Assay Description:
Inhibition against Aminopeptidase P from human platelets.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Xaa-Pro dipeptidase
(Homo sapiens (Human))
Pharmacia And Upjohn
Curated by
ChEMBL
Ligand
BDBM50078393
((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.30E+5nM
Assay Description:
Inhibition against Prolidase from pig kidney.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI