Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50395027(CHEMBL2163441)Copy SMILESCopy InChI

Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetEstrogen receptor [D538G](Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership

US Patent

LigandBDBM263244(US9708370, 45 CP-1B(iii))Copy SMILES

Affinity DataIC50:  1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL

LigandBDBM50395027(CHEMBL2163441)Copy SMILESCopy InChI

Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI