Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProlyl endopeptidase(Mus musculus)
University Of Helsinki

Curated by ChEMBL

LigandBDBM50529474(CHEMBL4528594)Copy SMILESCopy InChI

Affinity DataIC50:  91nMAssay Description:Inhibition of PREP in C57BL/6 mouse cortex homogenate assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-4-methylcoumarin as s...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProlyl endopeptidase(Sus scrofa)
University Of Helsinki

Curated by ChEMBL

LigandBDBM50529474(CHEMBL4528594)Copy SMILESCopy InChI

Affinity DataIC50:  129nMAssay Description:Inhibition of recombinant porcine brain PREP expressed in Escherichia coli assessed as formation of 7-amido-4-methylcoumarin using Suc-Gly-Pro-amido-...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
DrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI