Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sib Swiss Institute Of Bioinformatics

Curated by ChEMBL

LigandBDBM50465750(CHEMBL4292914)Copy SMILESCopy InChI

Affinity DataIC50:  282nMAssay Description:Antagonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as inhibition of ghrelin-induced intracellular calcium release inc...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sib Swiss Institute Of Bioinformatics

Curated by ChEMBL

LigandBDBM50465750(CHEMBL4292914)Copy SMILESCopy InChI

Affinity DataEC50:  117nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI