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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Mast/stem cell growth factor receptor Kit [D816V]
(Homo sapiens (Human))
Plexxikon
US Patent
Ligand
BDBM368753
(N-[(1S)-1-(3-chlorophenyl)ethyl]-2,2- dimethyl-4-[...)
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Affinity Data
Ki: 500nM
Assay Description:
The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Plexxikon
US Patent
Ligand
BDBM368753
(N-[(1S)-1-(3-chlorophenyl)ethyl]-2,2- dimethyl-4-[...)
Copy SMILES
Affinity Data
Ki: 5.50E+3nM
Assay Description:
The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI