Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
BDBM432966(5-cyclopropyl-N-((2S,4S)-1-(((R)-3,4- dimethylpipe...)
BDBM432996(5-cyclopropyl-N-((2S,4S)-1-((3,4- dimethylpiperazi...)
IC50: 193nMAssay Description:The assays were all performed in a buffer consisting of 25 mM Tris-Cl pH 8.0, 1 mM TCEP, 0.005% BSG, and 0.005% Tween 20, prepared on the day of use....More data for this Ligand-Target Pair
BDBM433032(5-cyclopropyl-N-((2S,4S)-1-(((S)-3,4- dimethylpipe...)
IC50: 446nMAssay Description:The assays were all performed in a buffer consisting of 25 mM Tris-Cl pH 8.0, 1 mM TCEP, 0.005% BSG, and 0.005% Tween 20, prepared on the day of use....More data for this Ligand-Target Pair