Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
IC50: 22nMAssay Description:Inhibition of human BACE2 using biotin-GLTNIKTEEISEISYEVEFR-C[Oregon green]KK-OH as substrate after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
IC50: 29nMAssay Description:Inhibition of human BACE1 using biotin-GLTNIKTEEISEISYEVEFR-C[Oregon green]KK-OH as substrate after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
IC50: 33nMAssay Description:Beta-secretase (BACE) is one of the enzymes involved in the generation of the amyloid beta peptide found in the amyloid plaques of Alzheimer's Di...More data for this Ligand-Target Pair
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)
BDBM223396(US9315520, 7 | US9315520, Example 7 | US9605007, E...)