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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
G-protein coupled estrogen receptor 1
(Homo sapiens (Human))
G1 Therapeutics
US Patent
Ligand
BDBM349624
((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
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Affinity Data
IC50: <1.00E+3nM
Assay Description:
A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Estrogen receptor
(Homo sapiens (Human))
G1 Therapeutics
US Patent
Ligand
BDBM349624
((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <1.00E+3nM
Assay Description:
All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences #IB00401. In an effort to screen selective es...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Estrogen receptor
(Homo sapiens (Human))
G1 Therapeutics
US Patent
Ligand
BDBM349624
((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <1.00E+3nM
Assay Description:
A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
G-protein coupled estrogen receptor 1
(Homo sapiens (Human))
G1 Therapeutics
US Patent
Ligand
BDBM349624
((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <1.00E+3nM
Assay Description:
All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences # IB00401. In an effort to screen selective e...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI