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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349624((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Affinity DataIC50: <1.00E+3nMAssay Description:A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349624((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Affinity DataIC50: <1.00E+3nMAssay Description:All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences #IB00401. In an effort to screen selective es...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEstrogen receptor(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349624((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Affinity DataIC50: <1.00E+3nMAssay Description:A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349624((S)-(4-fluoro-2,6-dimethylphenyl)(6- hydroxy-3-(4-...)
Affinity DataIC50: <1.00E+3nMAssay Description:All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences # IB00401. In an effort to screen selective e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent