Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 14 hits in this display
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
Ki: 650nMAssay Description:Inhibition of human HK1 using H-D-Val-Leu-Arg-AFC as substrate assessed as release of AFC after 10 to 120 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
BDBM189434(US9174974, Example 19)
Ki: 1.50E+3nMAssay Description:Inhibition of human plasmin using H-(D)-Val-Leu-LyspNA as substrate assessed as release of pNA after 10 to 120 mins by spectrophotometric methodMore data for this Ligand-Target Pair
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
Ki: 3.40E+3nMAssay Description:Inhibition of human factor 11a using pyroGlu-Pro-Arg-pNA as substrate assessed as release of pNA after 10 to 120 mins by spectrophotometric methodMore data for this Ligand-Target Pair
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
Ki: 7.50E+3nMAssay Description:Inhibition of human factor 12a using H-(D)-CHT-Gly-Arg-pNA as substrate assessed as release of pNA after 10 to 120 mins by spectrophotometric methodMore data for this Ligand-Target Pair
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
BDBM189434(US9174974, Example 19)
Ki: 1.50E+4nMAssay Description:Inhibition of human urokinase using pyro-Glu-Gly-Arg-pNA as substrate assessed as release of pNA after 10 to 120 mins by spectrophotometric methodMore data for this Ligand-Target Pair