Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5-hydroxytryptamine receptor 3A(RAT)
Virginia Commonwealth University

Curated by PDSP K_i Database

LigandBDBM50025470(2-Piperidin-1-yl-quinoline | CHEMBL76495 | N4-Deaz...)Copy SMILESCopy InChI

Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target5-hydroxytryptamine receptor 3A/3B/3C/3D/3E(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL

LigandBDBM50025470(2-Piperidin-1-yl-quinoline | CHEMBL76495 | N4-Deaz...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMAssay Description:Compound was tested for the inhibition of [3H]-GR-65,630 binding to 5-hydroxytryptamine 3 receptor expressed in NG 108-15 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaantibodypediaantibodypediaantibodypediaantibodypediaGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL

LigandBDBM50025470(2-Piperidin-1-yl-quinoline | CHEMBL76495 | N4-Deaz...)Copy SMILESCopy InChI

Affinity DataKi: >1.50E+5nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI