Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50256282((2R,2'R))-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)p...)
Affinity DataKi:  1.16E+4nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAchR in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50256282((2R,2'R))-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)p...)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed