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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300863
(3-[6-([3-[4-(3-Hydroxy-3- methylbutoxy)-2- methylp...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 16nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300872
((3S)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 500nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300873
((3R)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300863
(3-[6-([3-[4-(3-Hydroxy-3- methylbutoxy)-2- methylp...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 16nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300873
((3R)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300873
((3R)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300863
(3-[6-([3-[4-(3-Hydroxy-3- methylbutoxy)-2- methylp...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 16nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300872
((3S)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 500nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM300872
((3S)-3-(6-((3-(4-(3-Hydroxy-3- methylbutoxy)-2- me...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 500nM
Assay Description:
Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI