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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50344067
(CHEMBL1777860 | rac-3-(4-(2-methyl-4-(trifluoromet...)
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Affinity Data
IC50: 40nM
Assay Description:
Inhibition of human GPR40 expressed in CHO cells by SPA based binding assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50344067
(CHEMBL1777860 | rac-3-(4-(2-methyl-4-(trifluoromet...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 94nM
Assay Description:
Agonist activity at human GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Mus musculus)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50344067
(CHEMBL1777860 | rac-3-(4-(2-methyl-4-(trifluoromet...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 127nM
Assay Description:
Agonist activity at mouse GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI