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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProtein O-GlcNAcase(Homo sapiens (Human))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577841(CHEMBL4845911)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase(Bos taurus)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50577841(CHEMBL4845911)
Affinity DataKi:  3.00E+4nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed