Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 32 hits in this display
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
IC50: 370nMAssay Description:Inhibition of CDK1 in human MCF7 cells assessed as reduction in PP1alpha phosphorylation at T320 residue incubated for 6 hrs by immunoblot analysisMore data for this Ligand-Target Pair
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
IC50: >1.00E+4nMAssay Description:Inhibition of CDK2 in human MCF7 cells assessed as reduction in Rb phosphorylation at T821 residue incubated for 6 hrs by immunoblot analysisMore data for this Ligand-Target Pair
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
IC50: >1.00E+4nMAssay Description:Inhibition of CDK4/6 in human MCF7 cells assessed as reduction in Rb phosphorylation at S807/811 residue incubated for 6 hrs by immunoblot analysisMore data for this Ligand-Target Pair
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
Kd: 0.0894nMAssay Description:Binding affinity to human CDK9/CyclinT assessed as equilibrium dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
BDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)