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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 20nM
Assay Description:
Inhibition of BRD3-BD2 (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 71nM
Assay Description:
Inhibition of BRD2-BD2 (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 130nM
Assay Description:
Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.30E+3nM
Assay Description:
Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.70E+3nM
Assay Description:
Inhibition of BRD2-BD1 (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9.50E+3nM
Assay Description:
Inhibition of BRD3-BD1 domain (unknown origin) incubated for 6 hrs by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
Cnrs
Curated by
ChEMBL
Ligand
BDBM50586222
(CHEMBL5082786)
Copy SMILES
Copy InChI
Affinity Data
Kd: 150nM
Assay Description:
Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by ITC method
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI