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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetHistone deacetylase 2(Homo sapiens (Human))
The General Hospital

US Patent
LigandPNGBDBM592452(US11572368, Compound 140)
Affinity DataIC50:  555nMAssay Description:HDAC2: The following trypsin-coupled protocol and Caliper protocol described Herein was used to assay the compounds of the invention. HDAC2-Kinetic I...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
The General Hospital

US Patent
LigandPNGBDBM592452(US11572368, Compound 140)
Affinity DataIC50:  3.05E+3nMAssay Description:HDAC1: The following trypsin-coupled protocol and Caliper protocol described Herein was used to assay the compounds of the invention. Trypsin Coupled...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
The General Hospital

US Patent
LigandPNGBDBM592452(US11572368, Compound 140)
Affinity DataIC50:  1.76E+4nMAssay Description:HDAC3: The following trypsin-coupled protocol and Caliper protocol described Herein was used to assay the compounds of the invention. HDAC3-Kinetic I...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent