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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant Cathepsin C using H-Gly-Arg-AMC as substrate pretreated for 30 mins followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50:  70nMAssay Description:Inhibition of Cathepsin C in human U-937 cells using H-Gly-Phe-AFC as substrate pretreated for 1 hr followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50:  115nMAssay Description:Inhibition of Cathepsin C in human THP-1 cells using H-Gly-Phe-AFC as substrate pretreated for 1 hr followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProcathepsin L(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of human recombinant Cathepsin L using Z-Leu-Arg-AMC as substrate pretreated for 60 mins followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCathepsin B(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human recombinant Cathepsin B using Z-Leu-Arg-AMC as substrate pretreated for 60 mins followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCathepsin S(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human recombinant Cathepsin S using MCA-Arg-Pro-Lys-Pro-Val-Glu-NVAL-Trp-Arg-Lys-(DNP)-NH2 as substrate pretreated for 60 mins followed...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCathepsin K(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50605255(CHEMBL5186557)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human Cathepsin K using MCA-Arg-Pro-Lys-Pro-Val-Glu-NVAL-Trp-Arg-Lys-(DNP)-NH2 as substrate pretreated for 60 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails PubMed