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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  277nMAssay Description:Inhibition of human erythrocytes mu-calpain after 30 mins by fluorometric assay using pep1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of human liver cathepsin L after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of human liver cathepsin B after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by fluorometric assay using pep2 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50:  6.65E+4nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver cathepsin D after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed