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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetArginase(Plasmodium falciparum)
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of Plasmodium falciparum arginase using L-arginine as substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Institutes For Pharmaceutical Discovery

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataIC50:  3.43E+3nMAssay Description:Inhibition of human recombinant full length Arg1 using L-arginine as substrate assessed as urea level after 1 hr by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Institutes For Pharmaceutical Discovery

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataIC50:  5.07E+3nMAssay Description:Inhibition of human Arg2 by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Institutes For Pharmaceutical Discovery

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataKd:  880nMAssay Description:Binding affinity to human arginase 1 using L-arginine as substrate by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Institutes For Pharmaceutical Discovery

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataKd:  880nMAssay Description:Binding affinity to human Arg I assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed