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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Vu University Amsterdam
Ligand
BDBM22536
(1-[3-(1H-imidazol-4-ylmethyl)phenyl]-3,3-dimethylb...)
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Affinity Data
Ki: 6nM ΔG°: -46.9kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Histamine H3 receptor
(Homo sapiens (Human))
Vu University Amsterdam
Ligand
BDBM22536
(1-[3-(1H-imidazol-4-ylmethyl)phenyl]-3,3-dimethylb...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 32nM ΔG°: -42.8kJ/mole EC50: 79nM
pH: 7.4 T: 2°C
Assay Description:
Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI