Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
Ki: 4.30nMAssay Description:Displacement of [33P]-2MeS-ADP from human P2Y1 receptor expressed in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: 2.5nMAssay Description:Antagonist activity at P2Y1 receptor in washed human platelets assessed as 1 uM 2-methylthio-ADP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
IC50: 1.60E+3nMAssay Description:Antagonist activity at P2X1 receptor in HEK293 cells assessed as alpha, beta-methylene ATP-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
IC50: >2.00E+4nMAssay Description:Displacement of [33P]-2MeS-ADP from P2Y12 receptor (unknown origin) transfected in HEK293 cells after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair