Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Curasen Therapeutics

US Patent

LigandBDBM485867(US10947196, Compound 03-3)Copy SMILESCopy InChI

Affinity DataEC50: <10nMAssay Description:Compound preparation. Candidate beta-adrenergic compounds, dissolved to 10 mM in DMSO, were diluted in 1× stimulation buffer 1 (Cisbio Part #64SB1FDD...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Curasen Therapeutics

US Patent

LigandBDBM485867(US10947196, Compound 03-3)Copy SMILESCopy InChI

Affinity DataEC50:  55nMAssay Description:Compound preparation. Candidate beta-adrenergic compounds, dissolved to 10 mM in DMSO, were diluted in 1× stimulation buffer 1 (Cisbio Part #64SB1FDD...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI