Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 57 hits in this display
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 0.0230nMAssay Description:Displacement of [125I]-endothelin-1 from human recombinant ETA receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.0810nMAssay Description:Displacement of [125I]MIP-1alpha from human recombinant CCR1 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 0.170nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine A3 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.170nMAssay Description:Displacement of [125I]NDP-alpha -MSH from human recombinant MT1 receptor after 240 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.190nMAssay Description:Displacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.210nMAssay Description:Displacement of [3H]-SCH 23390 from human recombinant dopamine D1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.210nMAssay Description:Displacement of [125I]NDP-alpha -MSH from human recombinant MC4 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 0.25nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS1 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 0.430nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 0.470nMAssay Description:Displacement of [125I][Sar1,Ile8]-AT-II from human recombinant AT1 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 0.610nMAssay Description:Displacement of [3H]-DPCPX from human recombinant adenosine A1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 1.70nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 1.70nMAssay Description:Displacement of [3H]-imipramine from recombinant human 5-HT transporter after 60 mins by scintillation counting relative to controlMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 1.80nMAssay Description:Displacement of [3H]7-OH-DPAT from human recombinant dopamine D2S receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 2nMAssay Description:Binding affinity to recombinant human RORgammat transfected in human HEK293T cells incubated for 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 3.40nMAssay Description:Displacement of [3H]nisoxetine from recombinant human norepinephrine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
IC50: 4.90nMAssay Description:Displacement of [3H]nisoxetine from recombinant human dopamine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 9.20nMAssay Description:Displacement of [3H]-CGS 21680 from human recombinant adenosine A2A receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
IC50: 142nMAssay Description:Displacement of [125I]APT from human recombinant histamine H2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
EC50: 2.80nMAssay Description:Inverse agonist activity at RORgammat in human CD4 positive T cells assessed as inhibition of IL17A production in human Th17 cells after 1 hrMore data for this Ligand-Target Pair
BDBM392076(US10301272, Example 7/9)
BDBM392076(US10301272, Example 7/9)
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