Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM92336(Dipeptide nitrile, 10)
Ki: >330nMpH: 6.0Assay Description:Inhibition of human liver cathepsin B using Cbz-Arg-Arg-pNA as substrate at pH 6 incubated for 30 mins measured for 20 mins by photometrical analysisMore data for this Ligand-Target Pair
Cathepsin S(Homo sapiens (Human))Rheinische Friedrich-Wilhelms-Universitat Bonn
BDBM92336(Dipeptide nitrile, 10)
Procathepsin L(Bos taurus (bovine))Rheinische Friedrich-Wilhelms-Universitat Bonn
BDBM92336(Dipeptide nitrile, 10)
Ki: 900nM ΔG°: -35.9kJ/molepH: 6.0 T: 2°CAssay Description:Cathepsin enzyme activities were calculated from kinetic measurements performed by fluorimetric detection of the product 7-amino-4-methylcoumarin at ...More data for this Ligand-Target Pair
Papain(Carica papaya)Rheinische Friedrich-Wilhelms-Universitat Bonn
BDBM92336(Dipeptide nitrile, 10)
Cathepsin K(Homo sapiens (Human))Rheinische Friedrich-Wilhelms-Universitat Bonn
BDBM92336(Dipeptide nitrile, 10)
Ki: 6.30E+3nM ΔG°: -30.9kJ/molepH: 5.0 T: 2°CAssay Description:Cathepsin enzyme activities were calculated from kinetic measurements performed by fluorimetric detection of the product 7-amino-4-methylcoumarin at ...More data for this Ligand-Target Pair