Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL

LigandBDBM50240395(CHEMBL4071750)Copy SMILESCopy InChI

Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University of Traditional Chinese Medicine

Curated by ChEMBL

LigandBDBM50240387(CHEMBL4098760)Copy SMILESCopy InChI

Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI