Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50013915(CHEMBL1081913)
Affinity DataEC50:  6.30E+5nMAssay Description:Agonist activity at human GPR119 overexpressed in CHO cells assessed as stimulation of cAMP production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50013915(CHEMBL1081913)
Affinity DataEC50:  5.13E+3nMAssay Description:Agonist activity at GPR119 (unknown origin) by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50013915(CHEMBL1081913)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GPR119 receptor expressed in HEK293 cells after 30 mins by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed