Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed