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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Arachidonate 5-lipoxygenase-activating protein
(Homo sapiens (Human))
Merck Frosst Center For Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50080256
(3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(6-c...)
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Affinity Data
IC50: 8nM
Assay Description:
Measuring the affinity of leukotriene synthesis inhibitor for 5-lipoxygenase activating protein by using [125I]-L-691,831 as radioligand.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Arachidonate 5-lipoxygenase-activating protein/Polyunsaturated fatty acid 5-lipoxygenase
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50080256
(3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(6-c...)
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Copy InChI
Affinity Data
IC50: 110nM
Assay Description:
Human whole blood was stimulated with calcium ionophore (A23187) and LTB 4 measured by enzyme immunoassay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Arachidonate 5-lipoxygenase-activating protein/Polyunsaturated fatty acid 5-lipoxygenase
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50080256
(3-[3-tert-Butylsulfanyl-1-(4-chloro-benzyl)-5-(6-c...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.70E+4nM
Assay Description:
Human whole blood was stimulated with calcium ionophore (A23187) and LTB 4 measured by enzyme immunoassay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI