Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Calcium/calmodulin-dependent protein kinase type 1D
(Homo sapiens (Human))
University Of Nottingham
Curated by
ChEMBL
Ligand
BDBM50545575
(CHEMBL4648967 | US11530193, Example 3)
Copy SMILES
Copy InChI
Affinity Data
IC50: 399nM
Assay Description:
Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Calcium/calmodulin-dependent protein kinase type 1D
(Homo sapiens (Human))
University Of Nottingham
Curated by
ChEMBL
Ligand
BDBM50545575
(CHEMBL4648967 | US11530193, Example 3)
Copy SMILES
Copy InChI
Affinity Data
IC50: 429nM
Assay Description:
The following describes an ADP-Glo Kinase Assay, which measures the ADP formed from a kinase reaction; the ADP generated is converted into ATP and is...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
University Of Nottingham
Curated by
ChEMBL
Ligand
BDBM50545575
(CHEMBL4648967 | US11530193, Example 3)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human MLK3 using myelin basic protein as substrate in presence of [gamma-33P]-ATP by hotspot kinase assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dual specificity mitogen-activated protein kinase kinase 5
(Homo sapiens (Human))
University Of Nottingham
Curated by
ChEMBL
Ligand
BDBM50545575
(CHEMBL4648967 | US11530193, Example 3)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human MEK5 using ERK5 as substrate in presence of [gamma-33P]-ATP by hotspot kinase assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI