Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetADP-ribosylation factor 6(Human)
Navigen

US Patent

LigandBDBM50027961(CHEMBL3360257 | US10849901, Compound 126)Copy SMILESCopy InChI

Affinity DataIC50:  6.70nMAssay Description:The primary biochemical assay uses a fluorometric assay for monitoring the replacement of bound nucleotide with a fluorogenic GTP derivative bearing ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In DepthDetails US Patent
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TargetCytochrome b-c1 complex subunit 7(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL

LigandBDBM50027961(CHEMBL3360257 | US10849901, Compound 126)Copy SMILESCopy InChI

Affinity DataIC50: >2.00E+4nMAssay Description:Modulation of UQCRB in human HepG2 cells assessed as inhibition of HIF-1alpha for 4 hrs under 1%O2 by Western blot analysisMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI