Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158133(US9024044, 61 | US9227949, 61 | US9655879, 61)
BDBM158126(US9024044, 54 | US9227949, 54)
Ki: 1.53nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ...More data for this Ligand-Target Pair
BDBM158126(US9024044, 54 | US9227949, 54)
Ki: 1.53nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
Ki: 1.53nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Ki: 1.76nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
BDBM158126(US9024044, 54 | US9227949, 54)
Ki: 1.76nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
BDBM158126(US9024044, 54 | US9227949, 54)
Ki: 1.76nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (...More data for this Ligand-Target Pair