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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222166
(2-amino-N-((S)-2-benzyloxy-1-{1-[2-(3-phenyl-propy...)
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Affinity Data
Ki: 820nM
Assay Description:
Displacement of [125I]Ghrelin from human GHSR1a after 1 hr
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222166
(2-amino-N-((S)-2-benzyloxy-1-{1-[2-(3-phenyl-propy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 59nM
Assay Description:
Agonist activity at human GHS receptor expressed in H4 glioma cells assessed as intracellular calcium concentration by FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI