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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222164
((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
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Affinity Data
Ki: 200nM
Assay Description:
Displacement of [125I]Ghrelin from human GHSR1a after 1 hr
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222164
((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 200nM
Assay Description:
Agonist activity at human GHS receptor expressed in H4 glioma cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222164
((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 17nM
Assay Description:
Agonist activity at human GHS receptor expressed in H4 glioma cells assessed as intracellular calcium concentration by FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Growth hormone secretagogue receptor type 1
(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by
ChEMBL
Ligand
BDBM50222164
((S)-2-amino-N-(2-(benzyloxy)-1-(1-(3-phenylpropyl)...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 17nM
Assay Description:
Agonist activity at human GHS receptor expressed in H4 glioma cells assessed as intracellular calcium concentration by FLIPR assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI