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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetCaspase-3(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibitory concentration against caspase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibitory concentration of compound required against Caspase-3 enzyme compared to acylated dipeptidesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  5.85E+3nMAssay Description:Inhibition of caspase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  5.85E+3nMAssay Description:Inhibitory concentration of compound required against Caspase-1 enzyme compared to acylated dipeptidesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  6.81E+3nMAssay Description:Inhibitory concentration of compound required against Caspase-7 enzyme compared to acylated dipeptidesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  6.81E+3nMAssay Description:Inhibitory concentration against caspase-7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-6(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration required against caspase-6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-6(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration of compound required against Caspase-6 enzyme compared to acylated dipeptidesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory concentration against caspase-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-8(Homo sapiens (Human))
Idun Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119211(CHEMBL100933 | [(R)-3-((S)-2-Hydroxy-5-oxo-tetrahy...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory concentration of compound required against Caspase-8 enzyme compared to acylated dipeptidesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed