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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of Fibroblast activation protein alpha (seprase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolyl endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Quiescent cell prolyl dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human Potassium channel HERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Dipeptidylpeptidase IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Dipeptidylpeptidase VIIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed