Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
Caspase-3(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM314073(US10167313, Compound 71 | Z-Asp-(D,L Ala(2'-quinol...)
Caspase-7(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM314073(US10167313, Compound 71 | Z-Asp-(D,L Ala(2'-quinol...)
IC50: 8.90E+3nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-9(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM314073(US10167313, Compound 71 | Z-Asp-(D,L Ala(2'-quinol...)
IC50: >1.00E+4nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-1(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM314073(US10167313, Compound 71 | Z-Asp-(D,L Ala(2'-quinol...)
IC50: >1.00E+4nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair
Caspase-5(Homo sapiens (Human))Genesis Technologies
US Patent
BDBM314073(US10167313, Compound 71 | Z-Asp-(D,L Ala(2'-quinol...)
IC50: >1.00E+4nMAssay Description:Selectivity of compound 55, compound 63, compound 48, compound 57, compound 88 toward caspase-1 (pro-inflammatory group), caspase-5 (group I), caspas...More data for this Ligand-Target Pair