Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Trustees of Tufts College

US Patent

LigandBDBM609740(US11707539, Compound 6795)Copy SMILESCopy InChI

Affinity DataIC50:  8.90nMAssay Description:The purpose of this assay is to determine the IC50 of various inhibitors against recombinant human dipeptidyl peptidase IV (DPPIV), fibroblast activa...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Trustees of Tufts College

US Patent

LigandBDBM609741(US11707539, Compound 6795D)Copy SMILESCopy InChI

Affinity DataIC50:  17nMAssay Description:The purpose of this assay is to determine the IC50 of various inhibitors against recombinant human dipeptidyl peptidase IV (DPPIV), fibroblast activa...More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetProlyl endopeptidase(Homo sapiens (Human))
Trustees of Tufts College

US Patent

LigandBDBM609740(US11707539, Compound 6795)Copy SMILESCopy InChI

Affinity DataIC50:  5.52E+3nMAssay Description:The purpose of this assay is to determine the IC50 of various inhibitors against recombinant human dipeptidyl peptidase IV (DPPIV), fibroblast activa...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetProlyl endopeptidase(Homo sapiens (Human))
Trustees of Tufts College

US Patent

LigandBDBM609741(US11707539, Compound 6795D)Copy SMILESCopy InChI

Affinity DataIC50:  7.45E+3nMAssay Description:The purpose of this assay is to determine the IC50 of various inhibitors against recombinant human dipeptidyl peptidase IV (DPPIV), fibroblast activa...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Trustees of Tufts College

US Patent

LigandBDBM609741(US11707539, Compound 6795D)Copy SMILESCopy InChI

Affinity DataIC50: >1.00E+5nMAssay Description:The purpose of this assay is to determine the IC50 of various inhibitors against recombinant human dipeptidyl peptidase IV (DPPIV), fibroblast activa...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI