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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataKi:  0.730nMAssay Description:Competitive inhibition of human PREP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human PREP using Z-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of FAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DPP9 using H-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human FAP using Z-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Tufts University Sackler School Of Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50431227(CHEMBL2333024)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DPP8 using H-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed