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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetCoagulation factor XII(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  97nMAssay Description:Inhibition of human factor 12a using H-D-Pro-Phe-Arg-p-nitroanilide as chromogenic substrate assessed as liberation of p-nitroaniline measured every ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  157nMAssay Description:Inhibition of human factor 12a using H-D-Pro-Phe-Arg-p-nitroanilide as chromogenic substrate assessed as liberation of p-nitroaniline in presence of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human factor 10a using methoxycarbonyl-D-Nle-Gly-Arg-pNA as substrate measured after 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of plasma kallikrein (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Urokinase-type plasminogen activator (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50583792(CHEMBL5090804)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of factor 7a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed