Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 8.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 12nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 150nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 160nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.10E+3nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.60E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 8.50E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.20E+4nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.50E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.60E+5nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
BDBM50050528(Boronic acid derivative | CHEMBL63698 | US11096924...)
IC50: 1.10E+6nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair