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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetBeta-secretase 1(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50210578(CHEMBL242315 | H-(S)Glu-(S)Leu-Asp-(R)Leupsi [POOH...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human BACE1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50297711((4S)-4-[(2S)-2-[(2S)-3-{[(1R)-1-[(2S)-2-[(2S)-2-[(...)
Affinity DataIC50:  12nMAssay Description:Inhibition of full-domain of BACE1 expressed in HEK393 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 2(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50210578(CHEMBL242315 | H-(S)Glu-(S)Leu-Asp-(R)Leupsi [POOH...)
Affinity DataIC50:  12nMAssay Description:Inhibition of BACE2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50210578(CHEMBL242315 | H-(S)Glu-(S)Leu-Asp-(R)Leupsi [POOH...)
Affinity DataIC50:  28nMAssay Description:Inhibition of cathepsin D expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed