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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMicrotubule-associated protein tau(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50295169(CHEMBL4177337)
Affinity DataKd:  763nMAssay Description:Binding affinity to human Tau (1 to 441 residues) by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50295169(CHEMBL4177337)
Affinity DataKd:  23nMAssay Description:Binding affinity to human Keap1 (322 to 609 residues) by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed