Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128971(CHEMBL304669 | {(S)-1-[2-(4-Cyclohexyloxy-phenylam...)
Affinity DataIC50:  43nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128971(CHEMBL304669 | {(S)-1-[2-(4-Cyclohexyloxy-phenylam...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128971(CHEMBL304669 | {(S)-1-[2-(4-Cyclohexyloxy-phenylam...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed