Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128965(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-cyclohexy...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128965(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-cyclohexy...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50128965(1H-Indole-2-carboxylic acid {(S)-1-[2-(4-cyclohexy...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed