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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Amura Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134127(CHEMBL607122)
Affinity DataKi:  3.5nMAssay Description:Binding affinity against human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase B(Leishmania mexicana)
Amura Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134127(CHEMBL607122)
Affinity DataKi:  50nMAssay Description:Binding affinity against Leishmania mexicana cysteine peptidase B (CPB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Amura Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134127(CHEMBL607122)
Affinity DataKi:  93nMAssay Description:Binding affinity against cruzaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Amura Therapeutics

Curated by ChEMBL
LigandPNGBDBM50134127(CHEMBL607122)
Affinity DataKi:  434nMAssay Description:Binding affinity against cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed