Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Oryctolagus cuniculus (rabbit))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50150525(4-Methyl-2-(4''-piperazin-1-yl-biphenyl-3-ylamino)...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against humanized rabbit cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50150525(4-Methyl-2-(4''-piperazin-1-yl-biphenyl-3-ylamino)...)
Affinity DataIC50:  24nMAssay Description:Inhibitory concentration against human cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50150525(4-Methyl-2-(4''-piperazin-1-yl-biphenyl-3-ylamino)...)
Affinity DataIC50:  93nMAssay Description:Inhibitory concentration against human cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50150525(4-Methyl-2-(4''-piperazin-1-yl-biphenyl-3-ylamino)...)
Affinity DataIC50:  108nMAssay Description:Inhibitory concentration against human cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed